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A novel one-pot, three-component reaction for the synthesis of isocoumarin-condensed pyrazoles
Date
2011-03-30
Author
OZCAN, Sevil
Dengiz, Çağatay
DELIOMEROGLU, Murat K.
ŞAHİN, Ertan
BALCI, METİN
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The one-pot, three-component reaction of substituted homophthalic anhydrides with hydrazine in DMF as solvent and reactant, at reflux temperature, afforded isochromeno[3,4-c]pyrazole-5(2H)-one derivatives in high yields. The mechanism and roles of the substrates were investigated and it was found that cyclic hydrazides were formed as intermediates.
Subject Keywords
Organic Chemistry
,
Biochemistry
,
Drug Discovery
URI
https://hdl.handle.net/11511/36317
Journal
TETRAHEDRON LETTERS
DOI
https://doi.org/10.1016/j.tetlet.2011.01.114
Collections
Department of Chemistry, Article
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BibTeX
S. OZCAN, Ç. Dengiz, M. K. DELIOMEROGLU, E. ŞAHİN, and M. BALCI, “A novel one-pot, three-component reaction for the synthesis of isocoumarin-condensed pyrazoles,”
TETRAHEDRON LETTERS
, pp. 1495–1497, 2011, Accessed: 00, 2020. [Online]. Available: https://hdl.handle.net/11511/36317.